| Drug |
ka (min-1) |
Reference |
| Ciprofloxacin* |
0.019 |
Am. J. Med., 82 (1987) 146-53 |
| Amoxicillin |
0.017 |
Antimicrob. Agents Chemother.,
17 (1980) 199-202 |
| Ofloxacin |
0.070 |
Antimicrob. Agents Chemother.,
31 (1987) 156-60 |
| Lomefloxacin |
0.063 |
Antimicrob. Agents Chemother.,
34 (1990) 17-20 |
| Cefpodoxime
proxetil* |
0.011 |
Antimicrob. Agents Chemother.,
36 (1992) 126-31 |
| Ciprofloxacin* |
0.011 |
Antimicrob. Agents Chemother.,
40 (1996) 29-34 |
| Didanosine |
0.012-0.013 |
Antimicrob. Agents Chemother.,
40 (1996) 161-5 |
| Dapsone |
0.017 |
Antimicrob. Agents Chemother.,
40 (1996) 2743-8 |
| Rifabutin |
0.003 |
Antimicrob. Agents Chemother.,
42 (1998) 2017-23 |
| Pleconaril |
0.012 |
Antimicrob. Agents Chemother.,
43 (1999) 634-8 |
| Ethionamide |
0.006-0.008 |
Antimicrob. Agents Chemother.,
45 (2000) 810-14 |
| Theophylline* |
0.037 |
Asian Pac. J. Allergy Immunol.,
12 (1994) 137-45 |
| Theophylline* |
0.001 |
Biol. Pharm. Bull., 18 (1995)
1590-98 |
| Isoxicam/phenytoin |
0.006-0.019 |
Biopharm. Drug Dispos., 8 (1987)
57-61 |
| Alminoprofen |
0.047 |
Biopharm. Drug Dispos., 16
(1995) 627-34 |
| Selegiline |
0.010-0.026 |
Biopharm. Drug Dispos., 18
(1997) 665-80 |
| Roquinimex |
0.077-0.11 |
Biopharm. Drug Dispos., 20
(1999) 347-54 |
| Sotalol |
0.008-0.021 |
Br. J. Clin. Pharmacol., 45
(1998) 485-90 |
| Ibruprofen Lysinate |
0.025 |
Br. J. Clin. Pharmacol., 52
(2001) 387-98 |
| Tafenoquine |
0.012 |
Br. J. Clin. Pharmacol., 52
(2001) 663-70 |
| Strontium |
0.057 |
Calcif. Tissue Int., 47 (1990)
136-41 |
| Hydroxyurea |
0.049 |
Cancer Chemother. Pharmacol., 35
(1995) 417-22 |
| Strontium |
0.005 |
Clin. Chem., 35 (1989) 1911-4 |
| Bisoprolol |
0.007-0.012 |
Clin. Pharmacokinet., 17 (1989)
53-63 |
| Clinafloxacin |
0.019 |
Clin. Pharmacokinet., 40 (2001)
307-15 |
| Carbamazepine* |
0.004-0.014 |
Clin. Pharm., 6 (1987) 646-9 |
| Fleroxacin |
0.027-0.10 |
Clin. Pharmacol. Ther., 47
(1990) 618-28 |
| Carbamazepine* |
0.006 |
Clin. Pharmacol. Ther., 50
(1991) 10-15 |
| Carbamazepine/Fluoxitine* |
0.01 |
Clin. Pharmacol. Ther., 50
(1991) 10-15 |
| Alprazolam |
0.018 |
Clin. Pharmacol. Ther., 53
(1993) 521-28 |
| Tacrolimus |
0.075 |
Clin. Pharmacol. Ther., 57
(1995) 281-90 |
| Recainam |
0.029-0.083 |
Clin. Pharmacol. Ther., 57
(1995) 492-8 |
| Chlorzoxazone |
0.052 |
Clin. Pharmacol. Ther., 58
(1995) 498-505 |
| Thalidomide |
0.006-0.007 |
Clin. Pharmacol. Ther., 65
(1999) 483-90 |
| Cefpodoxime |
0.014 |
Drug Invest., 7 (1994) 221-33 |
| Ethanol* |
0.017-0.043 |
Eur. J. Clin. Pharmacol., 26 (1984) 619-26 |
| Caffeine* |
0.040-0.076 |
Eur. J. Clin. Pharmacol., 31 (1987) 595-600 |
| Probenecid |
0.007 |
Eur. J. Clin. Pharmacol., 32 (1987) 395-401 |
| Disopyramide |
0.009 |
Eur. J. Clin. Pharmacol., 32 (1987) 625-9 |
| Propranolol |
0.025 |
Eur. J. Clin. Pharmacol., 38 (1990) 133-7 |
| Caffeine* |
0.053 |
Eur. J. Clin. Pharmacol., 39 (1990) 63-9 |
| Sun 1165 |
0.037 |
Eur. J. Clin. Pharmacol., 40 (1991) 411-4 |
| Cefadroxil |
0.01-0.02 |
Eur. J. Clin. Pharmacol., 41 (1991) 179-83 |
| Tianeptine |
0.010 |
Eur. J. Clin. Pharmacol., 45 (1993) 173-9 |
| Acetazolamide |
0.014 |
Eur. J. Clin. Pharmacol., 54 (1998) 63-8 |
| Caffeine* |
0.031-0.048 |
Eur. J. Clin. Pharmacol., 55 (1999) 445-9 |
| Mibefradil |
0.045 |
Int. J. Clin. Pharmacol. Res., 18 (1998)
63-71 |
| Pilocarpine HCl |
0.048 |
Jpn. J. Clin. Pharmacol. Ther., 30 (1999)
423-33 |
| Etoposide phosphate |
0.028 |
J. Clin. Oncol., 14 (1996) 2020-30 |
| Diltiazem |
0.016 |
J. Clin. Pharmacol., 28 (1988) 477-80 |
| Pranoprofen |
0.033-0.055 |
J. Clin. Pharmacol., 29 (1989) 786-90 |
| Valproic Acid |
0.015-0.034 |
J. Clin. Pharmacol., 29 (1989) 1048-52 |
| Didanosine |
0.022 |
J. Clin. Pharmacol., 32 (1992) 242-7 |
| Atenolol* |
0.017 |
J. Clin. Pharmacol., 35 (1995) 268-74 |
| Digoxin |
0.065-0.068 |
J. Clin. Pharmacol., 36 (1996) 247-56 |
| Furosemide* |
0.0005 |
J. Clin. Pharmacol., 36 (1996) 257-64 |
| Beta-methyldigoxin |
0.026-0.092 |
J. Clin. Pharmacol., |
| D-xylose |
0.015 |
J. Lab Clin. Med., 112 (1988) 533-43 |
| Carbamazepine* |
0.007 |
J. Pharm. Sci., 75 (1986) 897-900 |
| Betaxolol |
0.017-0.02 |
J. Pharm. Sci., 80 (1991) 321-4 |
| Atenolol* |
0.002 |
J. Pharm. Sci., 87 (1998) 403-410 |
| Terbutaline |
0.005 |
J. Pharm. Sci., 87 (1998) 403-410 |
| Antipyrine |
0.08 |
J. Pharm. Sci., 87 (1998) 403-410 |
| Metoprolol |
0.02 |
J. Pharm. Sci., 87 (1998) 403-410 |
| Furosemide* |
0.039 |
J. Pharmacobiodyn., 10 (1987) 370-6 |
| Ethanol* |
0.027 |
Methods Find. Exp. Clin. Pharmacol., 7
(1985) 539-44 |
| Terfenadine |
0.047 |
Pharm. Res., 13 (1996) 832-838 |
| BMS-187745 |
0.010 |
Pharm. Res., 15 (1998) 1782-6 |
| N-acetylprocainamide |
0.006 |
Pharmacotherapy, 5 (1985) 11-5 |
| Ofloxacin |
0.038 |
Pharmacotherapy, 12 (1992) 88-92 |
| Zidovudine |
0.067 |
Pharmacotherapy, 12 (1992) 429-34 |
| Carbamazepine* |
0.007 |
Pharmacotherapy, 18 (1998) 273-81 |
| Valproic Acid |
0.002 |
Ther. Drug Monit., 19 (1997) 516-20 |
| Pyridostigmine |
0.004 |
Xenobiotica, 23 (1993) 1263-75 |